Nọmba Cas: 1115-70-4 Ụdị Molecular: C4H11N5

Ngwaahịa

Nọmba Cas: 1115-70-4 Ụdị Molecular: C4H11N5

Nkọwa dị mkpirikpi:

Nọmba Cas: 1115-70-4
Aha kemịkalụ:
Ụdị ihe omimi: C4H11N5
Synonyms: Hydrochloride, Glucophage, wdg.


Nkọwa ngwaahịa

Mkpado ngwaahịa

nkọwapụta ngwaahịa

Ebe Na-agbaze 233-236 ℃
Njupụta 1.48g/cm³
nchekwa okpomọkụ 15-30 ℃
solubility Na-agbaze n'ime mmiri, soluble na ethanol, na nke na-adịghị edozi na chloroform na benzene.
ngwa anya ọrụ +25.7 degrees (C=1, mmiri)
Ọdịdị ọcha crystalline ntụ ntụ

ngwaahịa pharmacology

Usoro ọgwụ ọgwụ molekụla nke ugbu a aghọtachaghị nke ọma.A maara na ọ na-eme ma ọ dịkarịa ala na imeju, na-ebelata gluconeogenesis (ya bụ mmepụta glucose) na ibelata nguzogide insulin.Ụfọdụ ọmụmụ egosila na nwere ike ịgbalite AMP activated protein kinase (AMPK), nke bụ otu n'ime usoro dị mkpa maka igbochi gluconeogenesis imeju na imeziwanye mmetụta insulin na ụzọ ntụgharị insulin.AMPK, dị ka protein kinase, na-arụ ọrụ dị mkpa ọ bụghị naanị na ụzọ mgbaàmà insulin, kamakwa na nguzozi ike zuru oke na glucose na metabolism abụba.Nnwale anụmanụ na ọmụmụ ụlọ ọgwụ egosila na nwere ike ibute mgbanwe dị ukwuu na nhazi nke fecal microbiota na ọrịa shuga, nke nwere ike ọ bụghị naanị na-enye aka na nzuzo na mmetụta nke glucagon dị ka peptide-1 (GLP-1), mana gosikwa na ọ na-eme ka mmetụta insulin dịkwuo mma. , nke bụkwa otu n'ime usoro dị mkpa nke mmetụta mgbochi ọrịa shuga 2.

ngwaahịa eji

Ekwesịrị iji ngwaahịa a na obere doses ma jiri nwayọ mụbaa dịka ọnọdụ onye ọrịa siri dị.Usoro izizi nke ngwaahịa a (mbadamba hydrochloride) na-abụkarị gram 0,5, ugboro abụọ n'ụbọchị;Ma ọ bụ 0.85 grams, otu ugboro n'ụbọchị;Were na nri.

Ojiji na usoro onunu ogwu

Ekwesịrị iji ngwaahịa a na obere doses ma jiri nwayọ mụbaa dịka ọnọdụ onye ọrịa siri dị.Usoro izizi nke ngwaahịa a (mbadamba hydrochloride) na-abụkarị gram 0,5, ugboro abụọ n'ụbọchị;Ma ọ bụ 0.85 grams, otu ugboro n'ụbọchị;Were na nri.

Metformin

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